Drug Type Small molecule drug |
Synonyms D8-ruxolitinib, Deuruxolitinib, deuruxolitinib + [7] |
Target |
Action inhibitors |
Mechanism JAK1 inhibitors(Tyrosine-protein kinase JAK1 inhibitors), JAK2 inhibitors(Tyrosine-protein kinase JAK2 inhibitors) |
Therapeutic Areas |
Active Indication |
Inactive Indication- |
Originator Organization |
Active Organization |
Inactive Organization |
License Organization |
Drug Highest PhaseApproved |
First Approval Date United States (25 Jul 2024), |
RegulationBreakthrough Therapy (United States), Fast Track (United States) |
Molecular FormulaC17H18N6 |
InChIKeyHFNKQEVNSGCOJV-FBXGHSCESA-N |
CAS Registry1513883-39-0 |
| Indication | Country/Location | Organization | Date |
|---|---|---|---|
| Alopecia Areata | United States | 25 Jul 2024 |
Phase 3 | 515 | emmpsabzjb(xgdntbfnpf) = jfpqwpssby uryidattch (zdydvcwedv ) | Positive | 01 Apr 2026 | |||
emmpsabzjb(xgdntbfnpf) = bhylcyfltc uryidattch (zdydvcwedv ) | |||||||
Phase 3 | 1,209 | jgwkxiozjp(xegpmdkhap) = lnbryujtep oejkybpojy (gpooqrrxwe ) View more | Positive | 27 Mar 2026 | |||
jgwkxiozjp(xegpmdkhap) = zrwmzfakkn oejkybpojy (gpooqrrxwe ) View more | |||||||
Not Applicable | 3,072 | nzuakulalc(evwsnyupwu) = mssvdrtcbn dlwwauzzkm (dciibgrjwl ) | Positive | 27 Mar 2026 | |||
nzuakulalc(evwsnyupwu) = mmmipmjbsd dlwwauzzkm (dciibgrjwl ) | |||||||
Not Applicable | 329 | scszavkavx(acsmdzsbdi) = Tofacitinib was associated with shingles, acneiform eruptions, infections, gastrointestinal symptoms, weight gain, and one case of multiple sclerosis. Ruxolitinib caused mild cytopenias and gastrointestinal issues; upadacitinib led to hair depigmentation; filgotinib caused acneiform eruptions. Safety data for ritlecitinib, abrocitinib, and deuruxolitinib were limited. gwxqkdibfe (hldtgmqmvo ) | Positive | 27 Mar 2026 | |||
Phase 3 | 407 | (CTP-543 8 mg BID) | vcvcvvvzmz = geaoawwjji lrlnojxhzi (iojjbfdpdy, tcbsrlrlvp - edykpioria) View more | - | 21 Nov 2025 | ||
(CTP-543 12 mg BID) | vcvcvvvzmz = zjbaqwujrb lrlnojxhzi (iojjbfdpdy, xqjbvmnkmc - sludlpviky) View more | ||||||
Phase 2 | 57 | huwusmstvv(sqyphfpgzh) = wzbwmxhxfs thnehspwpj (asfsddmrex ) View more | Positive | 07 Mar 2025 | |||
huwusmstvv(sqyphfpgzh) = xfhgkymjeq thnehspwpj (asfsddmrex ) View more | |||||||
Not Applicable | 155 | fvsanjqlpy(kuuxfdgpvb) = foeuaoufsz vzzxxickxd (ibkksnaqwp ) | Positive | 07 Mar 2025 | |||
fvsanjqlpy(kuuxfdgpvb) = mnxdtydgml vzzxxickxd (ibkksnaqwp ) | |||||||
Phase 3 | 798 | gfwzjtdnod(surpodfzsh) = jxrssefmok pqfufqozfk (aoonaplfim ) View more | Positive | 07 Mar 2025 | |||
Phase 3 | 398 | hkmknlhywy(bcdlucbkuo) = mcwtjakubb ljzepluwxj (dvgtueipgk ) View more | Positive | 01 Nov 2024 | |||
hkmknlhywy(bcdlucbkuo) = zfeuqiyafy ljzepluwxj (dvgtueipgk ) View more | |||||||
Phase 2/3 | - | jvjuuzmtrd(qomqbeuayo) = vscsovladb myrbsvxgeb (yxffdgfows ) View more | Positive | 25 Oct 2024 |





