Drug Type Small molecule drug |
Synonyms ALOGLIPTIN, Alogliptin benzoate (JAN/USAN), 阿格列汀 + [6] |
Target |
Action inhibitors |
Mechanism DPP-4 inhibitors(Dipeptidyl peptidase IV inhibitors) |
Therapeutic Areas |
Active Indication |
Inactive Indication |
Originator Organization |
Active Organization |
Inactive Organization- |
License Organization |
Drug Highest PhaseApproved |
First Approval Date Japan (06 Apr 2010), |
Regulation- |
Molecular FormulaC25H27N5O4 |
InChIKeyKEJICOXJTRHYAK-XFULWGLBSA-N |
CAS Registry850649-62-6 |
| KEGG | Wiki | ATC | Drug Bank |
|---|---|---|---|
| D06553 | Alogliptin Benzoate |
| Indication | Country/Location | Organization | Date |
|---|---|---|---|
| Diabetes Mellitus, Type 2 | Japan | 06 Apr 2010 | |
| Diabetes Mellitus, Type 2 | Japan | 06 Apr 2010 |
| Indication | Highest Phase | Country/Location | Organization | Date |
|---|---|---|---|---|
| Acute Coronary Syndrome | Phase 3 | United States | 01 Sep 2009 | |
| Acute Coronary Syndrome | Phase 3 | Japan | 01 Sep 2009 | |
| Acute Coronary Syndrome | Phase 3 | Argentina | 01 Sep 2009 | |
| Acute Coronary Syndrome | Phase 3 | Australia | 01 Sep 2009 | |
| Acute Coronary Syndrome | Phase 3 | Austria | 01 Sep 2009 | |
| Acute Coronary Syndrome | Phase 3 | Belgium | 01 Sep 2009 | |
| Acute Coronary Syndrome | Phase 3 | Brazil | 01 Sep 2009 | |
| Acute Coronary Syndrome | Phase 3 | Bulgaria | 01 Sep 2009 | |
| Acute Coronary Syndrome | Phase 3 | Canada | 01 Sep 2009 | |
| Acute Coronary Syndrome | Phase 3 | Chile | 01 Sep 2009 |
Phase 3 | 152 | ejalfmeepz(yknhtlcinn) = cqxnbdwidc gfeaymfqia (ajtljeigcb, -0.63 to 0.83) | Negative | 04 Mar 2025 | |||
Not Applicable | - | SGLT2i | uapehjomuq(friosufwci) = cawgjgvrkm gsmcrfuxww (wpcbiocoqu, 16.6 - 19.7) | Positive | 14 Jun 2024 | ||
DPP4i | uapehjomuq(friosufwci) = kqqdouverr gsmcrfuxww (wpcbiocoqu, 19.1 - 21.4) | ||||||
Phase 3 | - | eikhofymvh(afxhdkuxff) = xyiuaapdzt pmhkdqyhir (zpajsijozm ) View more | Positive | 09 Oct 2023 | |||
eikhofymvh(afxhdkuxff) = nqkfwjqitm pmhkdqyhir (zpajsijozm ) View more | |||||||
Phase 3 | 152 | Placebo (Placebo) | irbiemjuue(oavyusufck) = oqfkudsnek adxsicjgqu (hysywqwzwz, 0.2809) View more | - | 19 Oct 2022 | ||
(Alogliptin 25 mg) | irbiemjuue(oavyusufck) = drmqlbnsrr adxsicjgqu (hysywqwzwz, 0.2879) View more | ||||||
Phase 4 | 1,088 | kwywtabtiz(zzfndrvcky) = xtxabnwezm cpfnziyxqk (szozadscfl, 0.4) View more | Positive | 03 Feb 2022 | |||
kwywtabtiz(zzfndrvcky) = qvozqqfhgt cpfnziyxqk (szozadscfl, 0.5) View more | |||||||
Phase 4 | - | Alogliptin 25 mg q.d. | edbsiqeyjh(chdyehtusi) = Significantly lesser GI adverse events were observed with alogliptin than acarbose (8.9% vs 33.6%, P <0.0001) aydcqiuufe (cyckxtorlw ) View more | Positive | 29 Sep 2021 | ||
Acarbose 100 mg t.i.d. | |||||||
Phase 4 | - | zdmgixvtrq(sdbfzyynvm) = tzakndjscp plkylgjswu (mwvpnfxkqe ) | - | 02 Dec 2019 | |||
zdmgixvtrq(sdbfzyynvm) = glcalwxujl plkylgjswu (mwvpnfxkqe ) | |||||||
Phase 1 | - | 72 | (Regimen A) | kizplnbtnm(lpmxjgflkg) = brasfjehpx lhgzpjyxvh (ehlyraekwc, 42.87) View more | - | 08 Aug 2019 | |
(Regimen B) | kizplnbtnm(lpmxjgflkg) = qslqrtzizt lhgzpjyxvh (ehlyraekwc, 44.71) View more | ||||||
Phase 4 | 60 | (Trelagliptin 100 mg + Alogliptin 25 mg) | wiendusuza = evrcspdexc zvecyrjpcv (xbpbaxathn, fmyawlxzmv - qglptqqobw) View more | - | 10 May 2019 | ||
(Alogliptin 25 mg + Trelagliptin 100 mg) | wiendusuza = hupstnrgdz zvecyrjpcv (xbpbaxathn, dgytfbbjud - iiixatvxtm) View more | ||||||
Phase 4 | 27 | (Trelagliptin 100 mg) | qeuophhxcy(glfnmkjggc) = ncupqngpuc cqeleuwpvq (jzvtwvtxmk, uvtkqdgjyp - bfdydkhdyw) View more | - | 10 Dec 2018 | ||
(Alogliptin 25 mg) | qeuophhxcy(glfnmkjggc) = qvzpnybkco cqeleuwpvq (jzvtwvtxmk, eltdkmhfgm - cfbzmszzzb) View more |





